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(1R,2S,3R)-Aprepitant

Cat.No.:HY-172514

CASNo.:1185502-97-9

分?式:C??H??F?N?O?

分?量:534.43

作?靶点:NeurokininReceptor

作?通路:GPCR/GProtein;NeuronalSignaling

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性(1R,2S,3R)-Aprepitant(Compoundent-4)是?种竞争性的?神经激肽-1(NK-1)受体拮抗剂。(1R,2S,3R)-

Aprepitant有望?于癌症和术后恶?呕吐的研究[1]。

REFERENCES

[1].KulangiapparK,etal.Syntheticcommunications:aninternationaljournalforrapidcommunicationofsyntheticorganicchemistry[J].

SyntheticCommunications,2014,1(44):2494-2502.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

Forresearchuseonly.

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