Hotline:400-820-3792
Inhibitors?ScreeningLibraries?Proteins
www.MedChemE
AH6809(Standard)
Cat.No.:HY-10418R
CASNo.:33458-93-4
分?式:C??H??O?
分?量:298.29
作?靶点:ProstaglandinReceptor
作?通路:GPCR/GProtein
储存?式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
?物活性AH6809(Standard)是AH6809的分析标准品。本产品?于研究及分析应?。AH6809是?种EP和DP受体
的拮抗剂，对克隆的?类EP1，EP2，EP3-III和DP受体的Ki值分别为1217、1150、1597和1415nM，对?
?EP2受体的Ki值为350nM。
REFERENCES
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andrelatedanalogs.BiochimBiophysActa.2000Jan17;1483(2):285-93.
[2].KiriyamaM,et,al.LigandbindingspecificitiesoftheeighttypesandsubtypesofthemouseprostanoidreceptorsexpressedinChinese
hamsterovarycells.BrJPharmacol.1997Sep;122(2):217-24.
[3].WoodwardDF,et,al.6-Isopropoxy-9-oxoxanthene-2-carboxylicacid(AH6809),ahumanEP2receptorantagonist.BiochemPharmacol.
1995Nov9;50(10):1731-3.
[4].ZoccalKF,et,al.OpposingrolesofL