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RS-57067
Cat.No.:HY-171470
CASNo.:179382-91-3
分?式:C??H??ClN?O?
分?量:341.79
作?靶点:COX
作?通路:Immunology/Inflammation
储存?式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
?物活性RS-57067是?种COX-2抑制剂，Ki为16.9μM。RS-57067通过抑制COX-2减少前列腺素(如PGE2)的?成
，从?缓解炎症反应。RS-57067可?于炎症免疫疾病的研究[1]。
IC50TargetCOX-2
16.9μM(Ki)
REFERENCES
[1].SoOY,etal.ThedynamicsofprostaglandinHsynthases.Studieswithprostaglandinhsynthase2Y355Funmaskmechanismsoftime-
dependentinhibitionandallostericactivation.JBiolChem.1998Mar6;273(10):5801-7.
McePdfHeight
Caution:Producthasnotbeenfullyvalidatedformedicalapplications.
Forresearchuseonly.
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1/1MasterofBioactiveMolecules—您?边的抑制剂?师