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Inhibitors?ScreeningLibraries?Proteins

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PI3K-IN-56

Cat.No.:HY-171558

CASNo.:2633645-58-4

分?式:C??H??F?N?O?

分?量:631.61

作?靶点:PI3K;Akt

作?通路:PI3K/Akt/mTOR

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性PI3K-IN-56(Compound1)是?种具有?服活性、强效、选择性的不可逆磷酸肌苷激酶(PI3K)抑制剂。PI3K-

IN-56不可逆地阻断磷脂酰肌醇-3,4,5-三磷酸(PIP3)的产?和下游AKT信号通路。PI3K-IN-56有望?于PI3Kα

驱动的癌症的研究，如乳腺癌和卵巢癌[1]。

REFERENCES

[1].NeilSoninDHAWAN,etal.Crystallineformsandsaltsofapi3kinhibitorandmethodsofmakingandmethodsofusethereof.

WO2023179771A1.2023-09-28.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

Forresearchuseonly.

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1/1MasterofBioactiveMolecules—您?边的抑制剂?师