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Hotline:400-820-3792

Inhibitors?ScreeningLibraries?Proteins

www.MedChemE

NCG

Cat.No.:HY-173642

CASNo.:2768230-55-1

分?式:C??H??ClN?O?

分?量:382.8

作?靶点:Galactokinase

作?通路:MetabolicEnzyme/Protease

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性NCG是?种选择性半乳糖激酶(GALK1)抑制剂，对?和??重组GALK1的IC50分别为7.69μM

和13.67μM。NCG在10μM浓度下对GALK2和其他激酶?活性。NCG可?于经典

半乳糖?症的研究。

REFERENCES

[1].LiuL,etal.Structure-BasedOptimizationofSmallMoleculeHumanGalactokinaseInhibitors.JMedChem.2021Sep23;64(18):13551-

13571.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

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1/1MasterofBioactiveMolecules—您?边的抑制剂?师