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Diphenidol-d10hydrochloride

Cat.No.:HY-A0082S

Synonyms:Difenidolhydrochloride-d10

分?式:C??H??D??ClNO

分?量:355.97

作?靶点:Isotope-LabeledCompounds;SodiumChannel;mAChR

作?通路:Others;MembraneTransporter/IonChannel;GPCR/GProtein;

NeuronalSignaling

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性Diphenidol-d10(hydrochloride)(Difenidolhydrochloride-d10)是氘代标记的Diphenidol(hydrochloride).

Diphenidolhydrochloride(Difenidolhydrochloride)是?种?选择性的毒蕈碱M1-M4受体(muscarinicM1-

M4receptor)拮抗剂，具有抗?律失常活性。Diphenidolhydrochloride也是神经细胞电压门控离?通道(

Na+，K+，Ca2+)的有效?特异性阻滞剂。Diphenidolhydrochloride可?于抗眩晕、?吐的研究。

体外研究Stableheavyisotopesofhydrogen,carbon,andotherelementshavebeenincorporatedintodrugmolecules,

largelyastracersforquantitationduringthedrugdevelopmentprocess.Deuterationhasgainedattention

becauseofitspotentialtoaffectthepharmacoki