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ProteinkinaseinhibitorH-7dihydrochloride(Standard)
Cat.No.:HY-100983R
CASNo.:108930-17-2
分?式:C??H??Cl?N?O?S
分?量:364.29
作?靶点:PKC
作?通路:Epigenetics;TGF-beta/Smad
储存?式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
?物活性ProteinkinaseinhibitorH-7(dihydrochloride)(Standard)是ProteinkinaseinhibitorH-7(dihydrochloride)
的分析标准品。本产品?于研究及分析应?。ProteinkinaseinhibitorH-7dihydrochloride是?种有效的PKC
蛋?激酶C抑制剂。在100μM时,ProteinkinaseinhibitorH-7dihydrochloride完全抑制TPA(?肤肿瘤启
动?,12-O-tetradecanoylphorbol-13-acetate)和磷脂酶C诱导的ODC(鸟氨酸脱羧酶)[1]。
REFERENCES
[1].FischerSM,etal.Mediationofphorbolester-inducedoxidantgenerationinmurineepidermalcellsbyproteinkinaseC.ToxicolInVitro.
1989;3(3):195-9.
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