基本信息
文件名称:Protein-kinase-inhibitor-H-7-dihydrochloride-Standard-生命科学试剂-MCE.pdf
文件大小:466.87 KB
总页数:1 页
更新时间:2025-05-24
总字数:约2.13千字
文档摘要

Hotline:400-820-3792

Inhibitors?ScreeningLibraries?Proteins

www.MedChemE

ProteinkinaseinhibitorH-7dihydrochloride(Standard)

Cat.No.:HY-100983R

CASNo.:108930-17-2

分?式:C??H??Cl?N?O?S

分?量:364.29

作?靶点:PKC

作?通路:Epigenetics;TGF-beta/Smad

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性ProteinkinaseinhibitorH-7(dihydrochloride)(Standard)是ProteinkinaseinhibitorH-7(dihydrochloride)

的分析标准品。本产品?于研究及分析应?。ProteinkinaseinhibitorH-7dihydrochloride是?种有效的PKC

蛋?激酶C抑制剂。在100μM时,ProteinkinaseinhibitorH-7dihydrochloride完全抑制TPA(?肤肿瘤启

动?,12-O-tetradecanoylphorbol-13-acetate)和磷脂酶C诱导的ODC(鸟氨酸脱羧酶)[1]。

REFERENCES

[1].FischerSM,etal.Mediationofphorbolester-inducedoxidantgenerationinmurineepidermalcellsbyproteinkinaseC.ToxicolInVitro.

1989;3(3):195-9.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

Forresearchuseonly.

Tel:400-820-3792;021Fax:021E-mail:tech@MedChemE