Hotline:400-820-3792

Inhibitors?ScreeningLibraries?Proteins

www.MedChemE

Itopride-d6

Cat.No.:HY-B0732AS

CASNo.:1346746-82-4

Synonyms:HSR803-dfreebase

6

分?式:C??H??D?N?O?

分?量:364.47

作?靶点:Isotope-LabeledCompounds;DopamineReceptor;Bacterial;

Cholinesterase(ChE)

作?通路:Others;GPCR/GProtein;NeuronalSignaling;Anti-infection

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性Itopride-d6(HSR803-d6(freebase))是氘代标记的Itopride.Itopride(HSR803freebase)是?种?服有效的多

巴胺2(dopamine-2)拮抗剂和?酰胆碱酯酶(AChE)抑制剂。Itopride通过抗多巴胺能和抗?酰胆碱酯作?增

强胃动?，可?作胃肠促动?剂。Itopride可?于胃?管返流疾病(GERD)的研究。

体外研究Stableheavyisotopesofhydrogen,carbon,andotherelementshavebeenincorporatedintodrugmolecules,

largelyastracersforquantitationduringthedrugdevelopmentprocess.Deuterationhasgainedattention

becauseofitspotentialtoaffectthepharmacokineticandmetabolic