基本信息
文件名称:Macupatide-LY3532226-生命科学试剂-MCE.pdf
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更新时间:2025-06-12
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文档摘要

Hotline:400-820-3792

Inhibitors?ScreeningLibraries?Proteins

www.MedChemE

Macupatide

Cat.No.:HY-P10959

CASNo.:2923558-68-1

Synonyms:LY3532226

分?式:C???H???N??O??

分?量:4984.6

Sequence:Tyr-{Aib}-Glu-Gly-Thr-Phe-Ile-Ser-Asp-Tyr-Ser-Ile-{2-Me-Leu}-

Leu-Asp-Lys-{Lys-AEEA-AEEA-gGlu-C20diacid}-His-Gln-{Aib}

-Asp-Phe-Val-Glu-{pyridin-4-yl-Ala}-Leu-Leu-Glu-Ala-Gly-Pro-

Ser-Ser-Gly-Ala-Pro-Pro-Pro-Ser-NH2

SequenceShortening:Y-{Aib}-EGTFISDYSI-{2-Me-Leu}-LDK-{Lys-AEEA-AEEA-

gGlu-C20diacid}-HQ-{Aib}-DFVE-{pyridin-4-yl-Ala}-

LLEAGPSSGAPPPS-NH2

作?靶点:InsulinReceptor

作?通路:ProteinTyrosineKinase/RTK

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性Macupatide是?种抑胃肽(GIP)受体激动剂,可?于抗糖尿病的研究[1]。

REFERENCES

[1].WHO.InternationalNonproprietaryNamesforPharmaceuticalSubstances(INN),ProposedInternationalNonproprietaryNames:List

132.WHODrugInformation,Vol.38,No.4,2024.

McePdfHeight

Caution:Product