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Cbz-(S,S)-Pro-Pro-allyl
Cat.No.:HY-172790
分?式:C??H??N?O?
分?量:386.44
作?靶点:COX;Lipoxygenase
作?通路:Immunology/Inflammation;MetabolicEnzyme/Protease
储存?式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
?物活性Cbz-(S,S)-Pro-Pro-allyl(compound1a)是环氧合酶-2和5-脂氧合酶的双重抑制剂,对COX-1、COX-2和5-LOX
的IC50值分别为0.146nM、0.003nM和0.64nM。Cbz-(S,S)-Pro-Pro-allyl具有抗炎活性[1]。
REFERENCES
[1].ViveshVivesh,etal.ArationaleapproachindevelopingprolinebasedsmallpeptideasU-shapedanaloguesofarachidonicacid:Dual
inhibitorsofcyclooxygenase-2and5-lipoxygenasefordevelopinganti-inflammatoryagents.BioorgChem.2025Jun15:160:108452.
McePdfHeight
Caution:Producthasnotbeenfullyvalidatedformedicalapplications.
Forresearchuseonly.
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1/1MasterofBioactiveMolecules—您?边的抑制剂?师