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Inhibitors?ScreeningLibraries?Proteins
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CP-66713
Cat.No.:HY-111129
CASNo.:91896-57-0
分?式:C??H??ClN?
分?量:295.73
作?靶点:AdenosineReceptor
作?通路:GPCR/GProtein
储存?式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
?物活性CP-66713是?种选择性adenosineA2receptor拮抗剂，Ki为22nM。CP-66713可抑制诱发突触电位的长期
增强。CP-66713可?于神经系统疾病的研究[1]。
IC50TargetadenosineA2receptor:Kiof22nM
REFERENCES
[1].SekinoY,etal.Adenosine(A2)antagonistinhibitsinductionoflong-termpotentiationofevokedsynapticpotentialsbutnotofthe
populationspikeinhippocampalCA1neurons.BiochemBiophysResCommun.1991Dec31;181(3):1010-4.
McePdfHeight
Caution:Producthasnotbeenfullyvalidatedformedicalapplications.
Forresearchuseonly.
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