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Antidepressantagent10

Cat.No.:HY-W009754

CASNo.:87691-87-0

分?式:C??H??N?S

分?量:219.31

作?靶点:5-HTReceptor

作?通路:GPCR/GProtein;NeuronalSignaling

储存?式:RT,protectfromlight

*Insolvent:-80°C,6months;-20°C,1month(RT,protect

fromlight)

BIOLOGICALACTIVITY

?物活性Antidepressantagent10(Compound4)是?种具有?服活性的化合物。Antidepressantagent10对5-HT1A

和5-HT2受体的IC50分别为190nM和110nM。Antidepressantagent10可?于精神疾病的研究。

IC50Target5-HT1AReceptor5-HT2Receptor

190nM(IC50)110nM(IC50)

REFERENCES

[1].CipollinaJA,etal.Synthesisandbiologicalactivityoftheputativemetabolitesoftheatypicalantipsychoticagenttiospirone.JMed

Chem.1991Nov;34(11):3316-28.

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

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