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E3LigaseLigand-linkerConjugate163

Cat.No.:HY-170862

分?式:C??H??N?O?S

分?量:586.74

作?靶点:E3LigaseLigand-LinkerConjugates

作?通路:PROTAC

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性E3LigaseLigand-linkerConjugate163是AH078(HY-170859)的E3连接酶配体-连接?偶联物部分。AH078

是?种靶向降解CK1δ和CK1ε的PROTAC，可?于昼夜节律失调相关疾病的研究[1]。

REFERENCES

[1].HaagA,etal.DevelopmentandDiscoveryofaSelectiveDegraderofCaseinKinases1δ/ε.JMedChem.2025Jan9;68(1):506-530.

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Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

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