基本信息
文件名称:CDK2-IN-40-生命科学试剂-MCE.pdf
文件大小:457.61 KB
总页数:1 页
更新时间:2025-03-19
总字数:约1.9千字
文档摘要
Hotline:400-820-3792
Inhibitors?ScreeningLibraries?Proteins
www.MedChemE
CDK2-IN-40
Cat.No.:HY-170897
CASNo.:3065079-44-6
分?式:C??H??N?O?
分?量:343.38
作?靶点:CDK
作?通路:CellCycle/DNADamage
储存?式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
?物活性CDK9-IN-40是?种CDK2(Cyclindependentkinase2)抑制剂,详细信息请参考专利WO2024/254245A1
(Example1)。CDK9-IN-2抑制CDK2/CyclinE1的IC50为≤10nM。
IC50TargetCDK2/cyclinE
10nM(IC50)
REFERENCES
[1].HUMMELJoshua,etal.BICYCLICAMINESASCDK2INHIBITORS.WO2024/254245A1.WorldIntellectualPropertyOrganization.
12.12.2024
McePdfHeight
Caution:Producthasnotbeenfullyvalidatedformedicalapplications.
Forresearchuseonly.
Tel:400-820-3792;021Fax:021E-mail:tech@MedChemE
1/1MasterofBioactiveMolecules—您?边的抑制剂?师