基本信息
文件名称:CDK2-IN-40-生命科学试剂-MCE.pdf
文件大小:457.61 KB
总页数:1 页
更新时间:2025-03-19
总字数:约1.9千字
文档摘要

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Inhibitors?ScreeningLibraries?Proteins

www.MedChemE

CDK2-IN-40

Cat.No.:HY-170897

CASNo.:3065079-44-6

分?式:C??H??N?O?

分?量:343.38

作?靶点:CDK

作?通路:CellCycle/DNADamage

储存?式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

?物活性CDK9-IN-40是?种CDK2(Cyclindependentkinase2)抑制剂,详细信息请参考专利WO2024/254245A1

(Example1)。CDK9-IN-2抑制CDK2/CyclinE1的IC50为≤10nM。

IC50TargetCDK2/cyclinE

10nM(IC50)

REFERENCES

[1].HUMMELJoshua,etal.BICYCLICAMINESASCDK2INHIBITORS.WO2024/254245A1.WorldIntellectualPropertyOrganization.

12.12.2024

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

Forresearchuseonly.

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1/1MasterofBioactiveMolecules—您?边的抑制剂?师