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Dyrk1A-IN-12
Cat.No.:HY-170940
CASNo.:2243701-11-1
分?式:C??H??FN?O?S
分?量:405.44
作?靶点:DYRK;Enterovirus
作?通路:ProteinTyrosineKinase/RTK;Anti-infection
储存?式:Pleasestoretheproductundertherecommendedconditionsin
theCertificateofAnalysis.
BIOLOGICALACTIVITY
?物活性Dyrk1A-IN-12(compoundS43)是?种双特异性酪氨酸磷酸化调节激酶1A(Dyrk(Dualspecificitytyrosine
phosphorylationregulatedkinase1A)抑制剂。Dyrk1A-IN-12抑制Dyrk1A的IC50为95nM。Dyrk1A-IN-12
显?出抗EV-A71(肠道病毒A71)活性，其EC50为4.4μM，CC50为12.8μM，SI为2.9。Dyrk1A-IN-12对
单纯疱疹病毒(HSV)也表现出强效抑制作?。
IC50TargetDYRK1A
95nM(IC50)
McePdfHeight
Caution:Producthasnotbeenfullyvalidatedformedicalapplications.
Forresearchuseonly.
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1/1MasterofBioactiveMolecules—您?边的抑制剂?师